January 10, 2019

Dr. Elina Lidumniece

Researcher

E-mail: elinapetrova@osi.lv

Curriculum Vitae

Carrier Latvian Institute of Organic Synthesis, Riga, Latvia
Since 2023 Researcher
2015 Research Assistant
2014 Laboratory assistant

Department of Drug Design and Pharmacology, University of Copenhagen, Denmark
03.2022-05.2022 Visiting researcher
Education 2023 PhD, Riga Technical University, Faculty of Materials Science and Applied Chemistry
2015 
M.Sc. Chem., Faculty of Chemistry, University of Latvia
2013
 B.Sc. Chem., Faculty of Chemistry, University of Latvia
Awards2014-2015 “Olainfarm” Scholarship from University of Latvia foundation

Edit

List of Publications

4. Phenylglycinol Derived Chemistry

Lidumniece, E.; Bolsakova, J.; Grigorjeva, L. In Comprehensive Chirality, 2nd edition (Ed. J. R. Cossy). 2023, Accepted for publication Elsevier Inc. DOI:10.1016/B978-0-32-390644-9.00100-1

3. Subtilisin-like Serine Protease 1 (SUB1) as an Emerging Antimalarial Drug Target: Current Achievements in Inhibitor Discovery

Lidumniece, E.; Withers-Martinez, C.; Hackett, F.; Blackman, M. J.; Jirgensons, A. J. Med. Chem., 2022, 65, 12535-12545. DOI:10.1021/acs.jmedchem.2c01093

2. Peptidic boronic acids are potent cell-permeable inhibitors of the malaria parasite egress serine protease SUB1

Lidumniece, E.; Withers-Martinez, C.; Hackett, F.; Collins, C. R.; Perrin, A. J.; Koussis, K.; Bisson, C.; Blackman, M. J.; Jirgensons, A. Proc. Natl. Acad. Sci. U.S.A., 2021, 118, e2022696118. DOI:10.1073/pnas.2022696118



1. N-Sulfonylcarboxamide as an Oxidizing Directing Group for Ruthenium-Catalyzed C–H Activation/Annulation

Petrova, E.; Rasina, D.;  Jirgensons, A. Eur. J. Org. Chem., 2017, 1773-1779. DOI:10.1002/ejoc.201601582

Patents

  1. Jirgensons, A.; Lidumniece, E.; Withers-Martinez, C.; Blackman, M. J.; Finn, P. W.

WO2021/001697, A1, 07.01.2021